Probing Fluorinated Motifs onto Dual AChE-MAO B Inhibitors: Rational Design, Synthesis, Biological Evaluation, and Early-ADME Studies
2022-01-01 Rullo, M.; Cipolloni, M.; Catto, M.; Colliva, C.; Miniero, D. V.; Latronico, T.; De Candia, M.; Benicchi, T.; Linusson, A.; Giacche, N.; Altomare, C. D.; Pisani, L.
Thioxanthenone-based derivatives as multitarget therapeutic leads for Alzheimer's disease
2023-01-01 Tonelli, Michele; Catto, Marco; Sabaté, Raimon; Francesconi, Valeria; Laurini, Erik; Pricl, Sabrina; Pisani, Leonardo; Miniero, Daniela Valeria; Liuzzi, Grazia Maria; Gatta, Elena; Relini, Annalisa; Gavín, Rosalina; Del Rio, Jose Antonio; Sparatore, Fabio; Carotti, Angelo
The mitochondrial oxoglutarate carrier: from identification to mechanism
2013-01-01 Monné, M; Miniero, D; Iacobazzi, V; Bisaccia, F; Fiermonte, G.
Functional and structural role of amino acid residues in the even-numbered transmembrane alpha-helices of the bovine mitochondrial oxoglutarate carrier
2006-01-01 Cappello, Anna Rita; Curcio, Rosita; Valeria Miniero, Daniela; Stipani, Italo; Robinson, Alan J; Kunji, Edmund R S; Palmieri, Ferdinando
Neuroprotective Effect of Resveratrol against Manganese-Induced Oxidative Stress and Matrix Metalloproteinase-9 in an “In Vivo” Model of Neurotoxicity
2024-01-01 Latronico, Tiziana; Rossano, Rocco; Miniero, DANIELA VALERIA; Casalino, Elisabetta; Maria Liuzzi, Grazia
Mannich base approach to 5-methoxyisatin 3-(4-isopropylphenyl) hydrazone: a water-soluble prodrug for a multitarget inhibition of cholinesterases, beta-amyloid fibrillization and oligomer-induced cytotoxicity
2017-01-01 Pisani, Leonardo; DE PALMA, Annalisa; Giangregorio, Nicola; Miniero, DANIELA VALERIA; Pesce, Paolo; Nicolotti, Orazio; Campagna, Francesco; Altomare, Cosimo Damiano; Catto, Marco
Mitochondrial transporters for ornithine and related amino acids: A review
2015-01-01 Monné, Magnus; Miniero, DANIELA VALERIA; Daddabbo, Lucia; Palmieri, Luigi; Porcelli, Vito; Palmieri, Ferdinando
Chemical characterisation of PM10 from ship emissions: a study on samples from hydrofoil exhaust stacks
2022-01-01 Chianese, Elena; Tirimberio, Giuseppina; Appolloni, Luca; Dinoi, Adelaide; Contini, Daniele; Di Gilio, Alessia; Palmisani, Jolanda; Cotugno, Pietro; Miniero, Daniela Valeria; Dusek, Ulrike; Cammino, Gennaro; Riccio, Angelo
hERG stereoselective modulation by mexiletine‐derived ureas: Molecular docking study, synthesis, and biological evaluation
2023-01-01 Milani, Gualtiero; Budriesi, Roberta; Tavazzani, Elisa; Maddalena Cavalluzzi, Maria; Beatrice Mattioli, Laura; Miniero, DANIELA VALERIA; Delre, Pietro; Danilo Belviso, Benny; Denegri, Marco; Cuocci, Corrado; Paola Rotondo, Natalie; De Palma, Annalisa; Gualdani, Roberta; Caliandro, Rocco; Felice Mangiatordi, Giuseppe; Kumawat, Amit; Camilloni, Carlo; Priori, Silvia; Lentini, Giovanni
The mitochondrial oxoglutarate carrier: Cysteine-scanning mutagenesis of transmembrane domain IV and sensitivity of Cys mutants to sulfhydryl reagents
2001-01-01 Stipani, V.; Cappello, A. R.; Daddabbo, L.; Natuzzi, D.; Miniero, D. V.; Stipani, I.; Palmieri, F.
Citrate Regulates the Saccharomyces cerevisiae Mitochondrial GDP/GTP Carrier (Ggc1p) by Triggering Unidirectional Transport of GTP
2022-01-01 Seccia, R.; De Santis, S.; Di Noia, M. A.; Palmieri, F.; Miniero, D. V.; Marmo, R.; Paradies, E.; Santoro, A.; Pierri, C. L.; Palmieri, L.; Marobbio, C. M. T.; Vozza, A.
Substrate specificity of the two mitochondrial ornithine carriers can be swapped by single mutation in substrate binding site
2012-01-01 Monne, M.; Miniero, D. V.; Daddabbo, L.; Robinson, A. J.; Kunji, E. R. S.; Palmieri, F.
Substrate-induced conformational changes of the mitochondrial oxoglutarate carrier: A spectroscopic and molecular modelling study
2005-01-01 Della Rocca, B. M.; Miniero, D. V.; Tasco, G.; Dolce, V.; Falconi, M.; Ludovico, A.; Cappello, A. R.; Sanchez, P.; Stipani, I.; Casadio, R.; Desideri, A.; Palmieri, F.
Functional and Structural Role of Amino Acid Residues in the Odd-numbered Transmembrane α-Helices of the Bovine Mitochondrial Oxoglutarate Carrier
2007-01-01 Cappello, A. R.; Miniero, D. V.; Curcio, R.; Ludovico, A.; Daddabbo, L.; Stipani, I.; Robinson, A. J.; Kunji, E. R. S.; Palmieri, F.
Imaging Intron Evolution
2022-01-01 Antonietta Panaro, Maria; Calvello, Rosa; Miniero, DANIELA VALERIA; Mitolo, Vincenzo; Cianciulli, Antonia
Editorial: Understanding membrane transporters: from structure to function
2023-01-01 Pasquadibisceglie, A.; Bonaccorsi Di Patti, M. C.; Miniero, D. V.; Musci, G.; Polticelli, F.
Novel 6-alkyl-bridged 4-arylalkylpiperazin-1-yl derivatives of azepino[4,3-b]indol-1(2H)-one as potent BChE-selective inhibitors showing protective effects against neurodegenerative insults
2024-01-01 Samarelli, Francesco; Purgatorio, Rosa; Lopopolo, Gianfranco; Deruvo, Caterina; Catto, Marco; Andresini, Michael; Carrieri, Antonio; Nicolotti, Orazio; De Palma, Annalisa; Miniero, DANIELA VALERIA; de Candia, Modesto; Altomare, Cosimo D.
The interaction of hemin, a porphyrin derivative, with the purified rat brain 2-oxoglutarate carrier
2021-01-01 Miniero, D. V.; Spagnoletta, A.; Gambacorta, N.; Scalera, V.; Pierri, C. L.; Nicolotti, O.; De Palma, A.
Mitochondrial ATP-Mg/phosphate carriers transport divalent inorganic cations in complex with ATP
2017-01-01 Monné, M.; Daddabbo, L.; Giannossa, L. C.; Nicolardi, MARIA CRISTINA; Palmieri, L.; Miniero, D. V.; Mangone, A.; Palmieri, F.
Microwave-Assisted Extraction of Bioactive Compounds from Lentil Wastes: Antioxidant Activity Evaluation and Metabolomic Characterization
2022-01-01 Cavalluzzi, Maria Maddalena; Lamonaca, Antonella; Rotondo, Natalie Paola; Miniero, Daniela Valeria; Muraglia, Marilena; Gabriele, Paola; Corbo, Filomena; De Palma, Annalisa; Budriesi, Roberta; De Angelis, Elisabetta; Monaci, Linda; Lentini, Giovanni
| Titolo | Data di pubblicazione | Autore(i) | File |
|---|---|---|---|
| Probing Fluorinated Motifs onto Dual AChE-MAO B Inhibitors: Rational Design, Synthesis, Biological Evaluation, and Early-ADME Studies | 1-gen-2022 | Rullo, M.; Cipolloni, M.; Catto, M.; Colliva, C.; Miniero, D. V.; Latronico, T.; De Candia, M.; Benicchi, T.; Linusson, A.; Giacche, N.; Altomare, C. D.; Pisani, L. | |
| Thioxanthenone-based derivatives as multitarget therapeutic leads for Alzheimer's disease | 1-gen-2023 | Tonelli, Michele; Catto, Marco; Sabaté, Raimon; Francesconi, Valeria; Laurini, Erik; Pricl, Sabrina; Pisani, Leonardo; Miniero, Daniela Valeria; Liuzzi, Grazia Maria; Gatta, Elena; Relini, Annalisa; Gavín, Rosalina; Del Rio, Jose Antonio; Sparatore, Fabio; Carotti, Angelo | |
| The mitochondrial oxoglutarate carrier: from identification to mechanism | 1-gen-2013 | Monné, M; Miniero, D; Iacobazzi, V; Bisaccia, F; Fiermonte, G. | |
| Functional and structural role of amino acid residues in the even-numbered transmembrane alpha-helices of the bovine mitochondrial oxoglutarate carrier | 1-gen-2006 | Cappello, Anna Rita; Curcio, Rosita; Valeria Miniero, Daniela; Stipani, Italo; Robinson, Alan J; Kunji, Edmund R S; Palmieri, Ferdinando | |
| Neuroprotective Effect of Resveratrol against Manganese-Induced Oxidative Stress and Matrix Metalloproteinase-9 in an “In Vivo” Model of Neurotoxicity | 1-gen-2024 | Latronico, Tiziana; Rossano, Rocco; Miniero, DANIELA VALERIA; Casalino, Elisabetta; Maria Liuzzi, Grazia | |
| Mannich base approach to 5-methoxyisatin 3-(4-isopropylphenyl) hydrazone: a water-soluble prodrug for a multitarget inhibition of cholinesterases, beta-amyloid fibrillization and oligomer-induced cytotoxicity | 1-gen-2017 | Pisani, Leonardo; DE PALMA, Annalisa; Giangregorio, Nicola; Miniero, DANIELA VALERIA; Pesce, Paolo; Nicolotti, Orazio; Campagna, Francesco; Altomare, Cosimo Damiano; Catto, Marco | |
| Mitochondrial transporters for ornithine and related amino acids: A review | 1-gen-2015 | Monné, Magnus; Miniero, DANIELA VALERIA; Daddabbo, Lucia; Palmieri, Luigi; Porcelli, Vito; Palmieri, Ferdinando | |
| Chemical characterisation of PM10 from ship emissions: a study on samples from hydrofoil exhaust stacks | 1-gen-2022 | Chianese, Elena; Tirimberio, Giuseppina; Appolloni, Luca; Dinoi, Adelaide; Contini, Daniele; Di Gilio, Alessia; Palmisani, Jolanda; Cotugno, Pietro; Miniero, Daniela Valeria; Dusek, Ulrike; Cammino, Gennaro; Riccio, Angelo | |
| hERG stereoselective modulation by mexiletine‐derived ureas: Molecular docking study, synthesis, and biological evaluation | 1-gen-2023 | Milani, Gualtiero; Budriesi, Roberta; Tavazzani, Elisa; Maddalena Cavalluzzi, Maria; Beatrice Mattioli, Laura; Miniero, DANIELA VALERIA; Delre, Pietro; Danilo Belviso, Benny; Denegri, Marco; Cuocci, Corrado; Paola Rotondo, Natalie; De Palma, Annalisa; Gualdani, Roberta; Caliandro, Rocco; Felice Mangiatordi, Giuseppe; Kumawat, Amit; Camilloni, Carlo; Priori, Silvia; Lentini, Giovanni | |
| The mitochondrial oxoglutarate carrier: Cysteine-scanning mutagenesis of transmembrane domain IV and sensitivity of Cys mutants to sulfhydryl reagents | 1-gen-2001 | Stipani, V.; Cappello, A. R.; Daddabbo, L.; Natuzzi, D.; Miniero, D. V.; Stipani, I.; Palmieri, F. | |
| Citrate Regulates the Saccharomyces cerevisiae Mitochondrial GDP/GTP Carrier (Ggc1p) by Triggering Unidirectional Transport of GTP | 1-gen-2022 | Seccia, R.; De Santis, S.; Di Noia, M. A.; Palmieri, F.; Miniero, D. V.; Marmo, R.; Paradies, E.; Santoro, A.; Pierri, C. L.; Palmieri, L.; Marobbio, C. M. T.; Vozza, A. | |
| Substrate specificity of the two mitochondrial ornithine carriers can be swapped by single mutation in substrate binding site | 1-gen-2012 | Monne, M.; Miniero, D. V.; Daddabbo, L.; Robinson, A. J.; Kunji, E. R. S.; Palmieri, F. | |
| Substrate-induced conformational changes of the mitochondrial oxoglutarate carrier: A spectroscopic and molecular modelling study | 1-gen-2005 | Della Rocca, B. M.; Miniero, D. V.; Tasco, G.; Dolce, V.; Falconi, M.; Ludovico, A.; Cappello, A. R.; Sanchez, P.; Stipani, I.; Casadio, R.; Desideri, A.; Palmieri, F. | |
| Functional and Structural Role of Amino Acid Residues in the Odd-numbered Transmembrane α-Helices of the Bovine Mitochondrial Oxoglutarate Carrier | 1-gen-2007 | Cappello, A. R.; Miniero, D. V.; Curcio, R.; Ludovico, A.; Daddabbo, L.; Stipani, I.; Robinson, A. J.; Kunji, E. R. S.; Palmieri, F. | |
| Imaging Intron Evolution | 1-gen-2022 | Antonietta Panaro, Maria; Calvello, Rosa; Miniero, DANIELA VALERIA; Mitolo, Vincenzo; Cianciulli, Antonia | |
| Editorial: Understanding membrane transporters: from structure to function | 1-gen-2023 | Pasquadibisceglie, A.; Bonaccorsi Di Patti, M. C.; Miniero, D. V.; Musci, G.; Polticelli, F. | |
| Novel 6-alkyl-bridged 4-arylalkylpiperazin-1-yl derivatives of azepino[4,3-b]indol-1(2H)-one as potent BChE-selective inhibitors showing protective effects against neurodegenerative insults | 1-gen-2024 | Samarelli, Francesco; Purgatorio, Rosa; Lopopolo, Gianfranco; Deruvo, Caterina; Catto, Marco; Andresini, Michael; Carrieri, Antonio; Nicolotti, Orazio; De Palma, Annalisa; Miniero, DANIELA VALERIA; de Candia, Modesto; Altomare, Cosimo D. | |
| The interaction of hemin, a porphyrin derivative, with the purified rat brain 2-oxoglutarate carrier | 1-gen-2021 | Miniero, D. V.; Spagnoletta, A.; Gambacorta, N.; Scalera, V.; Pierri, C. L.; Nicolotti, O.; De Palma, A. | |
| Mitochondrial ATP-Mg/phosphate carriers transport divalent inorganic cations in complex with ATP | 1-gen-2017 | Monné, M.; Daddabbo, L.; Giannossa, L. C.; Nicolardi, MARIA CRISTINA; Palmieri, L.; Miniero, D. V.; Mangone, A.; Palmieri, F. | |
| Microwave-Assisted Extraction of Bioactive Compounds from Lentil Wastes: Antioxidant Activity Evaluation and Metabolomic Characterization | 1-gen-2022 | Cavalluzzi, Maria Maddalena; Lamonaca, Antonella; Rotondo, Natalie Paola; Miniero, Daniela Valeria; Muraglia, Marilena; Gabriele, Paola; Corbo, Filomena; De Palma, Annalisa; Budriesi, Roberta; De Angelis, Elisabetta; Monaci, Linda; Lentini, Giovanni |
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